明治薬科大学

薬化学研究室

2.　Transformation of Indole Alkaloids. VI. A Novel Conversion of Oxindole Alkaloids into Indole Alkaloids via Indoline Derivatives

Yamanaka E.; Saito N.; Suzuki Y.; Sakai S.
Chem. Pharm. Bull., 1982, 30, 2068-2078.

3.　Catalytic Hydrogenation of 7-Methoxy-6-methyl-8-nitro-1-isoquinolinecarbonitrile to Uncommon Products

Kubo A.; Saito N.; Nakahara S.; Iwata R.
Angew. Chem. Int. Ed. Engl., 1982, 94, 875-876.

4.　Isolation and Structural Elucidation of New Saframycins Y3, Yd-1, Yd-2, Ad-1, Y2b and Y2b-d

Yazawa K.; Takahashi K.; Mikami Y.; Arai T.; Saito N.; Kubo A.
J. Antibiot., 1986, 39, 1639-1650.

5.　Structure of Saframycin D, a New Dimeric Isoquinolinequinone Antibiotic

Kubo A.; Saito N.; Kitahara Y.; Takahashi K.; Yazawa K.; Arai T.
Chem. Pharm. Bull., 1987, 35, 440-442.

6.　Preparations and Reactions of (Z)-3-Arylidene-6-arylmethyl-2,5-piperazinediones Having Highly Oxygenated benzene Rings

Kubo A.; Saito N.; Yamato H.; Kawakami Y.
Chem. Pharm. Bull., 1897, 35, 2525-2532.

7.　A Promising Cyclization of the 3-Arylidene-6-arylmethyl-2,5-piperazinedione to Construct Tricyclic lactam as an Intermediate to Saframycin Synthesis.

TKubo A.; Saito N.; Nakamura M.; Ogata K.; Sakai S.
Heterocycles, 1986, 26, 1765-1770.

8.　Synthesis of Saframycins. I. Total Synthesis of (±)-Saframycin B and Its Congeners

Kubo A.; Saito N.; Yamauchi R.; Sakai S.
Chem. Pharm. Bull., 1987, 35, 2158-2161.

9.　A Facile Synthesis of 1,2,3,4-Tetrahydroisoquinolines Through Cyclization of O,N-Acetals

Kubo A.; Saito N.; Kawakami N.; Matsuyama Y.; Miwa T.
Synthesis, 1987, 824-827.

10.　A New Pigment from Streptomyces lavendulae

Mikami Y.; Takahashi K.; Fukushima K.; Yazawa K.; Arai T.; Kubo A.; Saito N.; Kawakami N.
J. Antibiot., 1987, 40, 385-387.

11.　Synthesis of Saframycins. II. Preparations and Reactions of N-Methyl-2,5- piperazinediones

Kubo A.; Saito N.; Yamato H.; Yamauchi R.; Hiruma K.; Inouye S.
Chem. Pharm. Bull., 1988, 36, 2607-2614.

12.　Stereoselective Total Synthesis of (±)-Saframycin B

Kubo A.; Saito N.; Yamato H.; Masubuchi K.; Nakamura M.
J. Org. Chem., 1988, 53, 4295-4310.

13.　Structural Stdies on Minor Componebts of Saframycin Group Antibiotic Saframycins F, G and H

Mikami Y.; Takahashi K.; Yazawa K.; Chen H. Y.; Arai A.; Kubo A.; Saito N.
J. Antibiot., 1988, 41, 734-740.

14.　A Facile Synthesis of 1,2,3,4-Tetrahydroisoquinolines Through Cyclization of O,N- Acetals. II. Syntheses of Isoquinolinequinone Antibiotics

Saito N.; Kawakami N.; Yamada E.; Kubo A.
Chem. Pharm. Bull., 1998, 37, 1493-1499.

15.　Synthesis of Saframycins. 3. Preparation of a Key Tricyclic Lactam Intermediate to Saframycin A

Saito N.; Yamauchi R.; Nishioka H.; Ida S.; Kubo A.
J. Org. Chem., 1989, 54, 5391-5395.

16.　Synthesis of Saframycins. IV. Selenium Oxide Oxidation of 4-Oxo-hexahydro-1,5-imino-3-benzazocin-7,10-dione: Promising Method to Construct Saframycins C and D from Saframycin B

Saito N.; Ōhira Y.; Kubo A.
Chem. Pharm. Bull., 1990, 38, 821-823.

17.　Synthesis of Saframycins. V. Selenium Oxide Oxidation of Hexahydro- 1,5-imino-3-benzazocine-7,10-dione: A Useful Method for Constructing Saframycins C and D from Saframycin B

Saito N.; Ōhira Y.; Wada N.; Kubo A.
Tetrahedron, 1990, 46, 7711-7728.

18.　A Toxic Substance Produced by Nocardia otitidiscaviarum Isolated from Cutaneous nocardiosis

Mikami Y.; Sen F.; Yazawa K.; Fukushima K.; Maeda A.; Uno J.; Terao K.; Saito N.; Kubo A.; Suzuki K.
Mycopathologia, 1990, 112, 113-118.

19.　Intractivation of Kinamycin A by Phosphorylation in Pathogenic Nocardia

Yazawa K.; Mikami Y.; Maeda A.; Kubo T.; Suzuki K.; Saito N.; Kubo A.
Microbiol. Immunol., 1991, 35, 39-48.

20.　The Useful Transformation of (－)-Saframycin A to (－)-Saframycin Mx Type Compound

Saito N.; Nishida M.; Kubo A.
Chem. Pharm. Bull., 1991, 39, 1343-1345.

21.　Synthesis of Saframycins. VII. The Synthesis of Novel Renieramycin Congeners

Saito N.; Yamauchi R.; Kubo A.
Heterocycles, 1991, 32, 1203-1214.

22.　Antigungal Activity of SL-1, a -Nitrostyrene Type Pigment and Its Synthetic Congeners

Mikami Y.; Yazawa K.; Maeda A.; Uno J.; Kubo A.; Saito N.; Kawakami N.
J. Antibiot., 1991, 44, 1454-1456.

23.　A Synthesis of 4-Cyanohexanydro-2H-benzo[b]quinolizine-7,10-dione as a Simple Model Compound of Saframycin A

Kubo A.; Nakai T.; Koizumi Y.; Saito N.; Mikami Y.; Yazawa K.; Uno J.
Heterocycles, 1992, 34, 1201-1211.

24.　Synthesis of Saframycins. VIII. Synthesis of the ABC Ring of Safracins

Saito N.; Obara Y.; Azumaya M.; Kubo A.
Chem. Pharm. Bull., 1992, 40, 2620-2626.

25.　Synthesis of Saframycins. IX. An Efficient Synthesis of the ABC Ring of Safracins

Saito N.; Obara Y.; Aihara T.; Harada S.; Shida Y.; Kubo A.
Tetrahedron, 1994, 50, 3915-3928.

26.　Acid Catalyzed Intramolecular Diels-Alder Reactions in Lithium Perchlorate-Diethyl Ether. Acid Promoted Migration of Terminally Restricted Substrate

Grieco P. A.; Beck J. P.; Handy S. T.; Saito N.; Daeuble J. F.
Tetrahedron Lett., 1994, 35, 6783-6787.

27.　Synthesis of Saframycins. X. Transformation of (－)-Saframycin A to (－)-Saframycin Mx Type Compound with the Structure Proposed for Saframycin E

Saito N.; Harada S.; Nishida M.; Inouye I.; Kubo A.
Chem. Pharm. Bull., 1995, 43, 777-782.

28.　Synthesis of Saframycins. XI. Synthetic Studies toward a Total Synthesis of Safracin A

Saito N.; Harada S.; Yamashita M.; Saito T.; Yamaguchi K.; Kubo A.
Tetrahedron, 1995, 51, 8213-8230.

29.　Synthesis of Saframycins. XII. Total Synthesis of (－)-N-Acetylsaframycin Mx 2 and its Epi-(+)-Enantiomer

Saito N.; Harada S.; Inouye I.; Yamaguchi K.; Kubo A.
Tetrahedron, 1995, 51, 8231-8246.

30.　A Synthesis of the Derivatives of 1,2,5,10,10a-Hexahydrobenz[f]indolizine-6,9-dione Having Antifungal Activity as a Simple Model of Saframycin A.

Kubo A.; Nakai T.; Koizumi Y.; Kitahara Y.; Saito N.; Mikami, Y.; Yazawa K.; Uno J.
Heterocycles, 1996, 42, 195-211.

31.　Carbocyclic Ring Construction via Intramolecular Ionic Diels-Alder Reactions in situ Generated Heteroatom-Stabilized Allyl Cations in High Polar Media

Grieco P. A.; Kaufman, M. G.; Daeuble, J. F.; Saito N.
J. Am. Chem. Soc., 1996, 118, 2095-2096.

32.　Synthetic Approaches toward Ecteinascidins. Part 1. Preparation of an (E)-2-Arylidene-3-benzyl-1,5-imino-3-benzazocin-4-one having a Protected Phenol in the E-Ring

Saito N.; Tashiro K.; Maru Y.; Yamaguchi K.; Kubo A.
J. Chem. Soc., Perkin Trans. 1., 1997, 53-69.

33.　Synthesis of Novel Octahydro-1,5-imino-4,7,10-trione Derivatives Having a Methyl Group at the C-2 Position as ABC Ring Models of Saframycins

Saito N.; Tanitsu M.; Betsui T.; Suzuki R.; Kubo A.
Chem. Pharm. Bull., 1997, 45, 1120-1129.

34.　Synthesis and Antitumor Evaluation of Octahydro-5-Hydroxy-1,5-inimo-3- benzazocin-4,7,10-triones

Saito N.; Sakai H.; Takai E.; Muranaka R.; Itabashi M.; Kubo A.
Heterocycles, 1997, 46, 309-320.

35.　An Improved Synthesis of the ABC Ring Model of Ecteinascidins.

Saito N.; Kamayachi H.; Tachi M.; Kubo A.
Heterocycles, 1999, 51, 9-12.

36.　A Concise Route to 3-Hydroxy-4-methoxy-5-methylbenzaldehyde Derivative

Saito N.; Tachi M.; Seki R.; Sugawara Y.; Takeuchi E.; Kubo A.
Synth. Commun., 2000, 30, 2407-2421.

37.　A Practical Synthesis of the ABC Ring Model of Ecteinascidins

Saito N.; Tachi M.; Seki R.; Kamayachi H.; Kubo A.
Chem. Pharm. Bull., 2000, 48, 1549-1557.

38.　Structure of Saframycin R

Saito N.; Kameyama N.; Kubo A.
Tetrahedron, 2000, 56, 9937-9944.

39.　13C NMR Spectral Assignment of 5-Hydroxy-1,5-imino-3-benzazocin-4,7,10-trione Derivatives: The Revised Structure of Renieramycin H

Saito N.; Sakai H.; Suwanborirux K.; Pummangura S.; Kubo A.
Heterocycles, 2001, 55, 21-28.

40.　Ecteinascidins 770 and 786 from the Thai Tunicate, Ecteinascidia sp

Suwanborirux K.; Charupant K.; Amnuoypol S.; Sunibhond P.; Kubo A.; Saito N.
J. Nat. Prod., 2002, 65, 935-937.

41.　Chemistry of Renieramycins. Part 2. Partial Reduction and Nucleophilic Substitution Hexahydro-1,5-imino-4-oxo-3-benzazocine-7,10-dione: Promising Method to Construct Renieramycin J from Renieramycin G via Renieramycin E

Koizumi Y.; Kubo A.; Suwanborirux K.; Saito N.
Heterocycles, 2002, 57, 2345-2355.

42.　Synthetic Approaches toward Ecteinascidins. Part 2. Preparation of the ABCDE Ring System of Ecteinascidins Having Characteristic Substituents in Both Benzene Rings

Saito N.; Seki R.; Kameyama N.; Sugimoto R.; Kubo A.
Chem. Pharm. Bull., 2003, 51, 821-831.

43.　Chemistry of Renieramycins. Part 3. Isolation and Structure of Stabilized Renieramycin Type Derivatives Possessing Antitumor Activity from Thai Sponge, Xestospongia Species Pretreated with Potassium Cyanide

Suwanborirux K.; Amnuoypol S.; Plubrukarn A.; Pummangura S.; Kubo A.; Tanaka C.; Saito N.
J. Nat. Prod., 2003, 66, 1441-1446.

44.　Chemistry of Antitumor Isoquinolinequinone Alkaloids: Unexpected Oxidative Degradation of Saframycin S to Generate Simple Isoquinoline Alkaloids, Mimosamycin and Mimocin

Saito N.; Koizumi Y.; Tanaka C.; Suwanborirux K.; Amnuoypol S.; Kubo A.
Heterocycles, 2003, 61, 79-86.

45.　Chemistry of Renieramycins. Part 4. Synthesis of a Simple Natural Marine Product, 6-Hydroxy-7-methoxyisoquinolinemethanol

Saito N.; Tanaka C.; Satomi T.; Oyama C.; Kubo A.
Chem. Pharm. Bull., 2004, 52, 282-286.

46.　Chemistry of Renieramycins. Part 5. Structure Elucidation of Renieramycin Type Derivatives O, Q, R, and S, from Thai marine Sponge, Xestospongia Species Pretreated with Potassium Cyanide

Amnuoypol S.; Suwanborirux K.; Pummangura S.; Kubo A.; Tanaka C.; Saito N.
J. Nat. Prod., 2004, 67, 1023-1028.

47.　Chemistry of Renieramycins. Part 6. Transformation of Renieramycin M into Jorumycin and Renieramycin J Including Oxidative Degradation Products, Mimosamycin, Renierone, and Renierol Acetate

Saito N.; Tanaka C.; Koizumi Y.; Suwanborirux K.; Amnuoypol S.; Pummangura S.; Kubo A.
Tetrahedron, 2004, 60, 3873-3881.

48.　Chemistry of Ecteinascidins. Part 2. Preparation of 6’-O-Acyl Derivatives of Stable Ecteinascidin and Evaluation of Cytotoxicity

Puthongking P.; Patarapanich C.; Amnuoypol S.; Suwanborirux K.; Kubo A.; Saito N.
Chem. Pharm. Bull., 2006, 54, 1010-1016.

49.　Synthesis of 1,2,3,4,5,6,7,10-Octahydro-1,5-imino-7,10-dioxo-3-benzazocine-4-carbonitrile Derivatives and Evaluation of Antitumor Activity Related to Saframycin and Renieramycin Isoquinolinequinones

Koizumi Y. Inamura K.; Kubo A.; Saito N.
Heterocycles, 2006, 70, 477-490.

50.　Jorunnamycins A-C, New Stabilized Renieramycin-Type Bistetrahydroisoquinolines Isolated from the Thai Nudibramch Jorunna funebris

Charupant K.; Suwanborirux K. Amnuoypol S.; Saito E.; Kubo A.; Saito N.
Chem. Pharm. Bull., 2007, 55, 81-86.

51.　Chemistry of Tetrahydroisoquinoline Antitumor Natural Products: Preparation and Antitumor Activity of Analogues of Cribrostatin 4

Saito E.; Daikuhara N.; Saito N.
Heterocycles, 2007, 74, 411-420.

52.　Synthesis of Tetrahydroisoquinoline Antitumor Natural Products: Construction of Tricyclic Lactams Through Pictet-Spengler-Type Cyclization of N-Methyl-3-Arylmethylpiperizine- 2,5-dione with Ethyl Diethoxyacetate

Yokoya M.; Kawachi O.; Saito N.
Heterocycles, 2008, 76, 1497-1509.

53.　JSPS Asia and Africa Scientific Platform Program: Development for the Medicinal Chemistry Based on Biologically Active Natural Products in the Subtropical Zone

Saito N.; Morita T.
Yakugaku Zasshi, 2009, 129, 407-412.

54.　Chemistry of Renieramycins. Part 7. Renieramycins T and U, Novel Renieramycin-Ecteinascidin Hybrid Marine Natural Products from Thai sponge, Xestospongia sp

Daikuhara N.; Tada Y.; Yamaki S.; Charupant K.; Amnuoypol S.; Suwanborirux K.; Saito N.
Tetrahedron Lett., 2009, 50, 4276-4278.

55.　Chemistry of Renieramycins. Part 8. Synthesis and Cytotoxicity Evaluation of Renieramycin M-Jorunamycin A Analogues

Charupant K.; Daikuhara N.; Saito E.; Amnuoypol S.; Suwanborirux K.; Owa T.; Saito N.
Bioorg. & Med. Chem., 2009, 17, 4548-4558.

56.　Microarray-based Transcriptional Profiling of Renieramycin M and Jorunnamycin C, Isolated from Thai Marine Organisms

Charupant K.; Suwanborirux K.; Daikuhara N.; Yokoya M.; Ushijima-Sugano, R.; Kawai T.; Owa T.; Saito N.
Marine Drugs, 2009, 7, 483-494.

57.　Chemistry of Renieramycins. Part 9: Stereocontrolled Total Synthesis of (±)-Renieramycin G

Yokoya M., Shinada-Fujino K., Saito N.
Tetrahedron Lett., 2011, 52, 2446-2449.

58.　Synthesis of Renieramycins: Construction of the Core Ring System of Cribrostatin 4 through Modified Pictet-Spengler Cyclization of 3,6-Bisarylpiperazine-2,5-dione with Diethoxyethyl Benzoate

Yokoya M., Ito H., Saito N.
Chem. Pharm. Bull., 2011, 59, 787-792.

59.　Chemistry of Ecteinascidins. Part 3. Preparation of 2’-N-Acyl Derivatives of Ecteinascidin 770 and Evaluation of Cytotoxicity

Saktrakulkla P., Toriumi S., Tsujimoto M., Patarapanich C., Suwanborirux K., Saito N.
Bioorig. Med. Chem., 2011, 19, 4421-4436. Corrigendum: 2012, 20, 531.

60.　Chemistry of Renieramycins. Part 11: Total Synthesis of (±)-Cribrostatin 4

Yokoya M., Ito H., Saito N.
Tetrahedron, 2011, 67, 9185-9192.

61.　Chemistry of Renieramycins. Part 10: Structure of Renieramycin V, A Novel Renieramycin Marine Natural Product Having a Sterol Ether at C-14 Position

Saito N., Yoshino M., Charupant K., Suwanborirux K.
Heterocycles, 2012, 84, 309-314.

62.　Molecular Network Profiling of U373MG Human Glioblastoma Cells Following Induction of Apoptosis by Novel Marine Derived Anti-Cancer 1,2,3,4-Tetrahydroisoquinoline Alkaloids

Tabunoki H., Saito N., Suwanborirux K., Charupant K., Satoh J.
Cancer Cell International, 2012, 12:14.

63.　Chemistry of Renieramycins. Part 12: An Improved Total Synthesis of (±)-Renieramycin G

Yokoya M., Shinada-Fujino K., Yoshida S., Mimura M., Takada H., Saito N.
Tetrahedron, 2012, 68, 4166-4181.

64.　Selenium Oxide Oxidation of Hexahydro-1,5-imino-3-benzazocine-7,10-dione in Aliphatic Alcohol for Conversion of Renieramycin Marine Natural Products

Mori M.; Daikuhara N.; Yamada J.; Saito N.
Heterocycles, 2012, 86, 317-330.

65.　Chemistry of Renieramycins. Part 13: Isolation and Structure of Stabilized Renieramycin Type Derivatives, Renieramycins W-Y, from Philippine Blue sponge Xestospongia sp., Pretreated with Potassium Cyanide

Tatsukawa M.; Punzalan L. L.; Magpantay H. D. S.; Villasenor I. M.; Concepcion G. P., Suwanborirux K.; Yokoya M.; Saito N.
Tetrahedron, 2012, 68, 7422-7428.

66.　Ecteinascidin 770, A Tetrahydroisoquinoline Alkaloid, Sensitizes Human Lung Cancer Cells to Anokis

Powan P.; Saito N.; Suwanborirux K.; Chanvorachote P.
Anticancer Res., 2013, 33, 505-512.

67.　Preparation of Tricyclic Lactam Model Compounds of Renieramycin and Saframycin Anticancer Natural Products from Common Intermediate

Nakai K.; Yokoya M.; Saito N.
Chem. Pharm. Bull., 2013, 61, 853-869.

68.　Replacement of a Quinone by a 5-O-Acetylhydroquinone Abolishes Accidental Necrosis-Inducing Effect while Preserving Apoptosis-Inducing Effect of Renieramycin M in Lung Cancer Cells

Cheun-Arom T.; Chanvorachote P.; Sirimangkalakitti N.; Chuanasa T.; Saito N.; Abe I.; Suwanborirux K.
J. Nat. Prod., 2013, 76, 1468-1474.

69.　Chemistry of Ecteinascidins. Part 4. Preparation of 2’-N-Acyl Ecteinascidin 770 analogues with Inproved Cytotoxicity Profile

Tsujimoto M.; Lowtangkitcharoen W.; Mori N.; Pangkruang W.; Puthongking P.; Suwanborirux K.; Saito N.
Chem. Pharm. Bull., 2013, 61, 1052-1064.

70.　Isolation, Structure Characterization, and Synthesis of Stabilized 1,2,3,4-Tetrahydroisoquinoline Marine Natural Product from Potassium Cyanide Pretreated Thai Tunicate, Ecteinascidia Thurstoni

Kimura S.; Pangkruang W.; Yokoya M.; Honda A.; Puthongking P.; Suwanborirux K.; Saito N.
Heterocycles, 2014, 88, 363-375.

71.　Preparation of Renieramycin Left-half Model Compounds

Nakai K.; Kubo K.; Yokoya M.; Saito N.
Tetrahedron, 2014, 70, 6529-6549.

72.　Synthetic Studies on Saframycin Antibiotics: An improved synthesis of tricyclic lactam intermediate and construction of the core ring system of saframycin A

Kimura S.; Kawai S.; Azuma M.; Umehara Y.; Koizumi Y.; Yokoya M.; Saito, N.
Heterocycles, 2015, 90, 327-343.

73.　Chemistry of Renieramycins. Part 14. Total Synthesis of Renieramycin I and Practical Synthesis of Cribrostatin 4 (Renieramycin H)

Yokoya M.; Kobayashi K.; Sato M.; Saito N.
Marine Drugs, 2015, 13, 4915-4933.

74.　Practical Synthesis of Tricyclic Lactam Model of Antitumor Renieramycin-Saframycin Natural Products

Yokoya M.; Fujino A.; Yaguchi K.; Yamazaki M.; Saito N.
Heterocycles, 2016, 93, 802-815.

75.　Synthesis and Absolute Configuration of Acanthodendrilline, a New Cytotoxic Bromotyrosine Alkaloid from Thai Marine Sponge Acanthodendrilla sp

Sirimangkalakitti N.; Yokoya M.; Chamni S.; Chanvorachote P.; Plubrukarn A.; Saito N.; Suwanborirux K.
Chem. Pharm. Bull., 2016, 64, 258-262.

76.　Stereoselective Total Synthesis of (-)-Renieramycin T

Yokoya M.; Toyoshima R.; Suzuki T.; Le V. H.; Williams R. M.; Saito N.
J. Org. Chem., 2016, 81, 4039-4047.

77.　Chemistry of Ecteinascidins. Part 5. An Additional Proof of Cytotoxicity Evaluation of Ecteinascidin 770 Derivatives

oyoshima R.; Mori N.; Suzuki T.; Lowtangkitcharoen W.; Suwanborirux K.; Saito N.
Chem. Pharm. Bull., 2016, 64, 966-969.

78.　Chemistry of Renieramycins. Part 15. Synthesis of 22-O-ester derivatives of Jorunnamycin A and their Cytotoxicity against Non-small Lung Cancer Cells

Sirimangkalakitti N.; Chamni S.; Charupant K.; Chanvorachote P.; Mori N.; Saito N.; Suwanborirux K.
J. Nat. Prod., 2016, 79, 2089-2093.

79.　Chemistry of Renieramycins. 16. Structure of 7-Desmethylrenieramycin O (= 14--Hydroxyrenieramycin S) from Blue Sponge, Xestospongia sp

Saito N.; Hiramatsu A.; Hirade H.; Kubota M.; Toyoshima R.; Fujino A.; Sirimangkalakitti N.; Suwanborirux K.; Concepcion G.
Heterocycles, 2017, 95, 748-752.

80.　Bishydroquinone Renieramycin M induced Human Lung Cancer Cell Apoptosis through Mitochondria-dependent Pathway

Pinkhien T.; Maiuthes A.; Chamni S.; Suwanborirux K.; Saito N.; Chanvorachote P.
Anticancer Res., 2016, 36, 6327-6333.

81.　Semisynthesis and Biological Evaluation of Prenylated Resveratrol Derivatives as Multi-Targeted Agents for Alzheimer’s Disease

Puksasook T.; Kimura S.; Tadtong S.; Jiaranakulwanitch J.; Pratungdejkul J.; Kitphati W.; Suwanborirux K.; Saito N.; Nukoolkarn V.
J. Nat. Med., 2017, 71 (4), 665-682.

82.　Chemistry of Renieramycins. 17. A New Generation of Renieramycins: 5-O-Ester Monohydroquinone Analogues of Renieramycin M as Potential Cytotoxic Agents against Non-Small-Cell Lung Cancer Cells

Chamni S.; Sirimangkalakitti N.; Chanvorachote P.; Saito N.; Suwanborirux K.
J. Nat. Prod., 2017, 80, 1541-1547.

83.　Apoptosis Inducing Effect of Hydroquinone-5-O-Cinnamoyl Ester Analog of Renieramycin M on Non-Small Cell Lung Cancer Cells

Maiuthed A.; Pinkhien T.; Chamni S.; Suwanborirux K.; Saito N.; Petpiroon N.; Chanvorachote P.
Anticancer Res., 2017, 37, 6259-6267.

84.　Preparation of Chiral Right-half Models of Antitumor Bistetrahydroisoquinoinequinone Natural Products

Senbonmatsu Y.; Kimura S.; Akiba M.; Ando S.; Saito N.
Heterocycles, 2018, 97, 1050-1067.

85.　A Stereocontrolled Total Synthesis of (±)-Saframycin A

Kimura S.; Saito N.
Tetrahedron, 2018, 74, 4504-4514.

86.　A Formal Synthesis of (+/-)-Renieramycin T

Kimura S.; Saito N.
ChemistryOpen, 2018, 7, 764-771.

87.　Synthesis of 6,6-Dimethyltricyclo[5.4.0.02,8]-Undecane-2,9-diol for (ent-)Longipinane-Type Sesquiterpenoids Using Two Types of Radical Cyclization

Matsunaga K.; Takatori K.: Kogen H.; Saito N.
Tetrahedron Lett., 2018, 59, 3872-3875.

88.　Preparation of Tricyclic Analog as CDE Ring Model of Renieramycin Marine Natural Product by Novel Photo-induced Transformation of 6-Methoxy-1,2,3,4-Tetrahydroisoquinline-5,8-dione

Yokoya M.; Takahashi S.; Saito N.
Heterocycles, 2019, 99, 1276-1303.

89.　Asymmetric Synthesis and Cytotoxicity Evaluation of Right-Half Models of Antitumor Renieramycin Marine Natural Products

Matsubara T.; Yokoya M.; Sirimangkalakitti N.; Saito N.
Marine Drugs, 2019, 17, 3

90.　5-O-Acetylrenieramycin T from Blue Sponge Xestospongia sp. induces Lung Cancer Stem Cells Apoptosis

Chantarawong W.; Chamni S.; Suwanborirux K.; Saito N.; Chanvorachote P.
Marine Drugs, 2019, 17, 109

91.　Naturally Occurring Biflavonoids with Amyloid- Aggregation Inhibitory Activity for Development of Anti-Alzheimer Agents

Sirimangkalakitti N.; Juliawaty L. D.; Hakim E. H.; Waliana J.; Saito N.; Koyama K.; Kinoshita K.
Bioorg. Med. Chem. Lett., 2019, 29, 1994-1997.

92.　Renieramycin T Induces Lung Cancer Cell Apoptosis by Targeting Mc-l-1 for Degradation: A New Insight in the Mechanism of Action

Petsri K.; Chamni S.; Suwanborirux K.; Saito N.; Chanvorachote P.
Marine Drugs, 2019, 17, 301.

93.　Synergistic Cytotoxicity of Renieramycin M (RM) and Doxorubicin (DOX) in MCF-7 Breast Cancer Cells

Tun J.; Salvador-Reyers L.; Velarde M.; Saito N.; Suwanborirux K.
Concepcion G. Marine Drugs, 2019, 17, 536.

94.　Total Synthesis of (+/-)-Marsupellines A and B via Acetoxymarsupelline Using a New Intramolecular Reductive Cyclization of Epoxy-cyanohydrin Derivative with CpZTiI

Matsunaga K.; Saito N.; Kogen H.; Takatori K.
Org. Lett., 2019, 21, 6054-6057.

95.　Chemistry of Renieramycins. Part 18. Synthesis of Renieramycin M and So-called Fennebricin A from (+/-)-Jorunnamycin A

Yokoya M.; Monden K.; Sato M.; Sirimangkalakitti N.; Saito N.
Heterocycles, 2020, 101, 548-558.

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